Journal of Postgraduate Medicine
 Open access journal indexed with Index Medicus & ISI's SCI  
Users online: 3277  
Home | Subscribe | Feedback | Login 
About Latest Articles Back-Issues Articlesmenu-bullet Search Instructions Online Submission Subscribe Etcetera Contact
 
Read this article

 


    Article Cited by others

SYMPOSIUM

Developing artemisinin based drug combinations for the treatment of drug resistant falciparum malaria: A review

Olliaro P L, Taylor W R

Year : 2004| Volume: 50| Issue : 1 | Page no: 40-44

   This article has been cited by
 
1 Modular synthesis and in vitro and in vivo antimalarial assessment of C-10 pyrrole Mannich base derivatives of artemisinin
Pacorel, B., Leung, S.C., Stachulski, A.V., Davies, J., Vivas, L., Lander, H., Ward, S.A., (...), OæNeill, P.M.
Journal of Medicinal Chemistry. 2010; 53(2): 633-640
[Pubmed]  [Google Scholar]
2 In vitro activity of mirincamycin (U24729A) against Plasmodium falciparum isolates from gabon
Held, J., Westerman, R., Kremsner, P.G., Mordmüller, B.
Antimicrobial Agents and Chemotherapy. 2010; 54(1): 540-542
[Pubmed]  [Google Scholar]
3 Design of a fixed-dose paediatric combination of artesunate and amodiaquine hydrochloride
Okwelogu, C., Clark, B., de Matas, M., Ifudu, D., Igwilo, C., Silva, B., York, P.
International Journal of Pharmaceutics. 2010; 387((1-2)): 19-25
[Pubmed]  [Google Scholar]
4 The effect of point mutations in dihydrofolate reductase genes and the multidrug resistance gene 1-86 on treatment of falciparum malaria in Sudan
Yusuf, R.U., Omar, S.A., Ngure, R.M.
Journal of Infection in Developing Countries. 2010; 4(2): 61-69
[Pubmed]  [Google Scholar]
5 Interaction of artemisinins with oxyhemoglobin Hb-FeII, Hb-FeII, carboxyHb-FeII, Heme-FeII, and carboxyheme FeII: Significance for mode of action and implications for therapy of cerebral malaria
Coghi, P., Basilico, N., Taramelli, D., Chan, W.-C., Haynes, R.K., Monti, D.
ChemMedChem. 2009; 4(12): 2045-2053
[Pubmed]  [Google Scholar]
6 Simple and rapid micro-scale quantification of artemisinin in living Artemisia annua L. by improved gas chromatography with electron-capture detection
Liu, S., Tian, N., Li, J., Huang, J., Liu, Z.
Biomedical Chromatography. 2009; 23(10): 1101-1107
[Pubmed]  [Google Scholar]
7 Malaria and iron: History and review Malaria and iron Eugene D. Weinberg and Jym Moon
Weinberg, E.D., Moon, J.
Drug Metabolism Reviews. 2009; 41(4): 644-662
[Pubmed]  [Google Scholar]
8 Discovery, mechanisms of action and combination therapy of artemisinin
Cui, L., Su, X.-Z.
Expert Review of Anti-Infective Therapy. 2009; 7(8): 999-1013
[Pubmed]  [Google Scholar]
9 Development of transgenic Artemisia annua (Chinese worm-wood) plants with an enhanced content of artemisinin, an effective anti-malarial drug, by hairpin-RNA-mediated gene silencing
Zhang, L., Jing, F., Li, F., Li, M., Wang, Y., Wang, G., Sun, X., Tang, K.
Biotechnology and Applied Biochemistry. 2009; 52(3): 199-207
[Pubmed]  [Google Scholar]
10 Building a golden triangle for the production and use of artemisinin derivatives against falciparum malaria in Africa
Brisibe, E.A., Uyoh, E.A., Brisibe, F., Magalhäes, P.M., Ferreira, J.F.S.
African Journal of Biotechnology. 2008; 7(25): 4884-4896
[Pubmed]  [Google Scholar]
11 Interplay between malaria, crystalline hemozoin formation, and antimalarial drug action and design
Weissbuch, I., Leiserowitz, L.
Chemical Reviews. 2008; 108(11): 4899-4914
[Pubmed]  [Google Scholar]
12 Artemisinin - An innovative cornerstone for anti-malaria therapy
Thomas, K., Ying, W.
Progress in Drug Research. 2008; 66: 383-422
[Pubmed]  [Google Scholar]
13 High efficacy of two artemisinin-based combinations (artemether- lumefantrine and artesunate plus amodiaquine) for acute uncomplicated malaria in Ibadan, Nigeria
Falade, C.O., Ogundele, A.O., Yusuf, B.O., Ademowo, O.G., Ladipo, S.M.
Tropical Medicine and International Health. 2008; 13(5): 635-643
[Pubmed]  [Google Scholar]
14 Making a difference: 30 years of TDR
Ridley, R.G., Fletcher, E.R.
Nature Reviews Microbiology. 2008; 6(5): 401-407
[Pubmed]  [Google Scholar]
15 Selective plasma protein binding of antimalarial drugs to α1-acid glycoprotein
Zsila, F., Visy, J., Mády, G., Fitos, I.
Bioorganic and Medicinal Chemistry. 2008; 16(7): 3759-3772
[Pubmed]  [Google Scholar]
16 Determination of artemisinin by post-column derivatization high performance liquid chromatography
Li, M., Wu, X., Yang, Y., Lin, H., Chai, Y., Hua, L.A.
Asian Journal of Chemistry. 2008; 20(3): 1907-1914
[Pubmed]  [Google Scholar]
17 The rapid determination of artemisinin by post-column derivatization high-performance liquid chromatography using matrix solid-phase dispersion method
Liu, H., Li, Q., Li, S., Zou, Y., Gu, A.
Journal of Chromatographic Science. 2008; 46(2): 122-126
[Pubmed]  [Google Scholar]
18 High efficacy of two artemisinin-based combinations (artemether-lumefantrine and artesunate plus amodiaquine) for acute uncomplicated malaria in Ibadan, Nigeria
Falade CO, Ogundele AO, Yusuf BO, et al.
TROPICAL MEDICINE & INTERNATIONAL HEALTH. 2008; 13(5): 635-643
[Pubmed]  [Google Scholar]
19 Timeline - Making a difference: 30 years of TDR
Ridley RG, Fletcher ER
NATURE REVIEWS MICROBIOLOGY. 2008; 6(5): 401-407
[Pubmed]  [Google Scholar]
20 Selective plasma protein binding of antimalarial drugs to alpha(1)-acid glycoprotein
Zsila F, Visy J, Mady G, et al.
BIOORGANIC & MEDICINAL CHEMISTRY. 2008; 16(7): 3759-3772
[Pubmed]  [Google Scholar]
21 Quantification of artemisinin in Artemisia annua extracts by H-1-NMR
Castilho PC, Gouveia SC, Rodrigues AI
PHYTOCHEMICAL ANALYSIS. 2008; 19(4): 329-334
[Pubmed]  [Google Scholar]
22 First assessment in humans of the safety, tolerability, pharmacokinetics, and ex vivo pharmacodynamic antimalarial activity of the new artemisinin derivative artemisone
Nagelschmitz J, Voith B, Wensing G, et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY. 2008; 52(9): 3085-3091
[Pubmed]  [Google Scholar]
23 Preparation of N-sulfonyl- and N-carbonyl-11-azaartemisinins with greatly enhanced thermal stabilities: in vitro antimalarial activities
Haynes RK, Wong HN, Lee KW, et al.
CHEMMEDCHEM. 2007; 2 (10): 1464-1479
[Pubmed]  [Google Scholar]
24 The Fe2+-mediated decomposotion, PfATP6 binding, and antimalarial activities of artemisone and other arteminisins: The unlikehood of C-centered radicals as bioactive intermediates
Haynes RK, Chan WC, Lung CM, et al.
CHEMMEDCHEM. 2007; 2 (10): 1480-1497
[Pubmed]  [Google Scholar]
25 A randomised controlled trial to assess the efficacy of dihydroartemisinin-piperaquine for the treatment of uncomplicated falciparum malaria in Peru
Grande T, Bernasconi A, Erhart A, et al.
PLOS CLINICAL TRIALS. 2007; 2 (10): Art. e1101
[Pubmed]  [Google Scholar]
26 Chemical instability determines the biological action of the artemisinins
Jansen FH, Soomro SA
CURRENT MEDICINAL CHEMISTRY. 2007; 14(30): 3243-3259
[Pubmed]  [Google Scholar]
27 Artesunate and dihydroartemisinin (DHA): Unusual decomposition products formed under mild conditions and comments an the fitness of DHA as an antimalarial drug
Haynes RK, Ho-Wai CM, Lung CM, et al.
CHEMMEDCHEM. 2007; 2 (10): 1448-1463
[Pubmed]  [Google Scholar]
28 Pumping iron: a potential target for novel therapeutics against schistosomes
Glanfield A, McManus DP, Anderson GJ, et al.
TRENDS IN PARASITOLOGY. 2007; 23 (12): 583-588
[Pubmed]  [Google Scholar]
29 An update on malaria prevention, diagnosis and treatment for the returning traveller
Gkrania-Klotsas E, Lever AML
BLOOD REVIEWS. 2007; 21 (2): 73-87
[Pubmed]  [Google Scholar]
30 Efficacy of sulfadoxine-pyrimethamine, amodiaquine, and sulfadoxine-pyrimethamine-amodiaquine combination for the treatment of uncomplicated falciparum malaria in the urban and suburban areas of Brazzaville (Congo)
Ndounga, M., Mayengue, P.I., Tahar, R., Casimiro, P.N., Matondo Maya, D.W., Miakassissa-Mpassi, V., Malonga, D.A., (...), Ntoumi, F.
Acta Tropica. 2007; 103(3): 163-171
[Pubmed]  [Google Scholar]
31 Artemisinin, promising lead natural product for various drug developments
Lee, S.
Mini-Reviews in Medicinal Chemistry. 2007; 7(4): 411-422
[Pubmed]  [Google Scholar]
32 Different doses of amodiaquine and chloroquine for treatment of uncomplicated malaria in children in Guinea-Bissau: implications for future treatment recommendations
Kofoed PE, Ursing J, Poulsen A, et al.
TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE. 2007; 101 (3): 231-238
[Pubmed]  [Google Scholar]
33 Amodiaquine and artemether-lumefantrine select distinct alleles of the Plasmodium falciparum mdr1 gene in Tanzanian children treated for uncomplicated malaria
Humphreys GS, Merinopoulos I, Ahmed J, et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY. 2007; 51 (3): 991-997
[Pubmed]  [Google Scholar]
34 Crystal nucleation, growth, and morphology of the synthetic malaria pigment beta-hematin and the effect thereon by quinoline additives: The malaria pigment as a target of various antimalarial drugs
Solomonov I, Osipova M, Feldman Y, et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY. 2007; 129 (9): 2615-2627
[Pubmed]  [Google Scholar]
35 Enoyl reductases as targets for the development of anti-tubercular and anti-malarial agents
Oliveir JS, Vasconcelos IB, Moreira IS, et al.
CURRENT DRUG TARGETS. 2007; 8 (3): 399-411
[Pubmed]  [Google Scholar]
36 A simple and efficient procedure to enhance artemisinin content in Artemisia annua L. by seeding to salinity stress
Qian, Z., Gong, K., Zhang, L., Lv, J., Jing, F., Wang, Y., Guan, S., (...), Tang, K.
African Journal of Biotechnology. 2007; 6(12): 1410-1413
[Pubmed]  [Google Scholar]
37 Prevalence of UGT1A9 and UGT2B7 nonsynonymous single nucleotide polymorphisms in West African, Papua New Guinean, and North American populations
Mehlotra RK, Bockarie MJ, Zimmerman PA
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY. 2007; 63 (1): 1-8
[Pubmed]  [Google Scholar]
38 Artemisinins for schistosomiasis and beyond
Utzinger J, Xiao SH, Tanner M, et al.
CURRENT OPINION IN INVESTIGATIONAL DRUGS. 2007; 8 (2): 105-116
[Pubmed]  [Google Scholar]
39 Lack of impact of artesunate on the disposition kinetics of sulfadoxine/pyrimethamine when the two drugs are concomitantly administered
Minzi OMS, Gupta A, Haule AF, et al.
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY. 2007; 63 (5): 457-462
[Pubmed]  [Google Scholar]
40 Inhibitors of de novo folat enzymes in Plasmodium falciparum
Nzila A
DRUG DISCOVERY TODAY. 2006; 11 (19-20): 939-944
[Pubmed]  [Google Scholar]
41 The efficacies of artesunate-sulfadoxine-pyrimethamine and artemether-lumefantrine in the treatment of uncomplicated, Plasmodium falciparum malaria, in an area of low transmission in central Sudan
Mohamed AO, Eltaib EH, Ahmed OA, Elamin SB, Malik EM
ANNALS OF TROPICAL MEDICINE AND PARASITOLOGY. 2006; 100 (1): 5-10
[Pubmed]  [Google Scholar]
42 Artemisone - A highly active antimalarial drug of the artemisinin class
Haynes RK, Fugmann B, Stetter J, et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION. 2006; 45 (13): 2082-2088
[Pubmed]  [Google Scholar]
43 From artemisinin to new artemisinin antimalarials: Biosynthesis, extraction, old and new derivatives, stereochemistry and medicinal chemistry requirements
Haynes RK
CURRENT TOPICS IN MEDICINAL CHEMISTRY. 2006; 6 (5): 509-537
[Pubmed]  [Google Scholar]
44 Prevalence of CYP2B6 alleles in malaria-endemic populations of West Africa and Papua New Guinea
Mehlotra RK, Ziats MN, Bockarie MJ, et al.
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY. 2006; 62 (4): 267-275
[Pubmed]  [Google Scholar]
45 Quantitation of artemisinin and its biosynthetic precursors in Artemisia annua L. by high performance liquid chromatography - electrospray quadrupole time-of-flight tandem mass spectrometry
Van Nieuwerburgh FCW, Casteele SRV, Maes L, et al.
JOURNAL OF CHROMATOGRAPHY A. 2006; 1118 (2): 180-187
[Pubmed]  [Google Scholar]
46 No hearing loss associated with the use of artemether-lumefantrine to treat experimental human malaria
McCall MBB, Beynon AJ, Mylanus EAM, et al.
TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE. 2006; 100 (12): 1098-1104
[Pubmed]  [Google Scholar]
47 Utility of alkylaminoquinolinyl methanols as new antimalarial drugs
Dow GS, Heady TN, Bhattacharjee AK, et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY. 2006; 50 (12): 4132-4143
[Pubmed]  [Google Scholar]
48 Current perspectives on the mechanism of action of artemisinins
Golenser J, Waknine JH, Krugliak M, et al.
INTERNATIONAL JOURNAL FOR PARASITOLOGY. 2006; 36 (14): 1427-1441
[Pubmed]  [Google Scholar]
49 Quantitation of artemisinin and its biosynthetic precursors in Artemisia annua L. by high performance liquid chromatography-electrospray quadrupole time-of-flight tandem mass spectrometry
Van Nieuwerburgh, F.C.W., Vande Casteele, S.R.F., Maes, L., Goossens, A., Inzé, D., Van Bocxlaer, J., Deforce, D.L.D.
Journal of Chromatography A. 2006; 1118(2): 180-187
[Pubmed]  [Google Scholar]
50 Malaria in the post-genomics era: light at the end of the tunnel or just another train?
Gardiner DL, McCarthy JS, Trenholme KR
POSTGRADUATE MEDICAL JOURNAL. 2005; 81 (958): 505-509
[Pubmed]  [Google Scholar]
51 Comparative efficacy of antimalarial drugs including ACTs in the treatment of uncomplicated malaria among children under 5 years in Ghana
Koram KA, Abuaku B, Duah N, Quashie N
ACTA TROPICA. 2005; 95 (3): 194-203
[Pubmed]  [Google Scholar]
52 Artemisinins
Woodrow, C.J., Haynes, R.K., Krishna, S.
Postgraduate Medical Journal. 2005; 81(952): 71-78
[Pubmed]  [Google Scholar]
53 Review: artesunate added to standard drug treatment reduces treatment failure in malaria
Garner P, Fanning MM
Evid Based Med. 2004; 9(5): 150
[HTML Full text] | [PDF]  [Google Scholar]
54 Falciparum malaria: Current therapeutic challenges
Maitland, K., Makanga, M., Williams, T.N.
Current Opinion in Infectious Diseases. 2004; 17(5): 405-412
[Pubmed]  [Google Scholar]
55 Artemisinins: Mechanisms of action and potential for resistance
Krishna S, Uhlemann AC, Haynes RK
Drug Resistance Updates. 2004; 7((4-5)): 233-244
[Pubmed]  [Google Scholar]
56 Association of house spraying with suppressed levels of drug resistance in Zimbabwe
Mharakurwa S, Mutambu SL, Mudyiradima R, Chimbadzwa T, Chandiwana SK, Day KP
Malar J. 2004; 3(1): 35
[Pubmed] | [PDF]  [Google Scholar]
57 In vitro sensitivity of Plasmodium falciparum to lumefantrine in north-western Thailand
Pilz JB, Wernsdorfer G, Sirichaisinthop J, et al.
WIENER KLINISCHE WOCHENSCHRIFT. 2004; 116((4 SUPPL)): 41-46
[Pubmed]  [Google Scholar]
58 Emerging drug - resistance and guidelines for treatment of malaria
M.Aslam Khan, Raymond A.smego Jr, Syed Tabish Razi, M. Asim Beg
Journal of the College of Physicians & Surgeons Pakistan. 2004; 14(5): 319-324
[Pubmed] | [PDF]  [Google Scholar]

 

Online since 12th February '04
© 2004 - Journal of Postgraduate Medicine
Official Publication of the Staff Society of the Seth GS Medical College and KEM Hospital, Mumbai, India
Published by Wolters Kluwer - Medknow